Acepromazine-d6 (maleaat)

Acepromazine-d6 (maleate) (Acetopromazine-d6 (maleate) ) is deuterium labeled Acepromazine (maleate) . Acepromazine (Acetopromazine) maleate is a phenothiazine tranquilizer and is alpha-adrenoceptor antagonist[1][2.

1331655-50-5

Acetopromazine-d6 (maleate) ; Acetylpromazine-d6 (maleate)

12352005

Adrenergic Receptor; Isotope-Labeled Compounds

GPCR/G Protein; Neuronal Signaling; Others

Neurological Disease

10 mM in DMSO

OC(/C=C/C(O)=O)=O.[2H]C([2H])([2H])N(C([2H])([2H])[2H])CCCN1C2=CC(C(C)=O)=CC=C2SC3=CC=CC=C31

C23H20D6N2O5S

448.56

[1]Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53 (2) :211-216.|[2]Gaulier JM, et al. Identification of acepromazine in hair: an illustration of the difficulties encountered in investigating drug-facilitated crimes. J Forensic Sci. 2008;53 (3) :755-759. |[3]Watney GC, et al. Effects of xylazine and acepromazine on bronchomotor tone of anaesthetised ponies. Equine Vet J. 1988;20 (3) :185-188.

Room temperature

http://file.medchemexpress.com/batch_PDF/HY-B1506AS/

Isotope-Labeled Compounds

No Development Reported