
ARV-771
Kwaliteit
ISO Gecertificeerd
Levering
24-48 uur
Technische Specificaties
1949837-12-0
C13474-1mg
PROTAC
Others
CC1=C (SC2=C1C (=NC (C3=NN=C (N32) C) CC (=O) NCCOCCCOCC (=O) NC (C (=O) N4CC (CC4C (=O) NC (C) C5=CC=C (C=C5) C6=C (N=CS6) C) O) C (C) (C) C) C7=CC=C (C=C7) Cl) C
C49H60ClN9O7S2
ARV-771 is a potent pan- (bromodomain and extra-terminal) BET degrader, a novel BET-PROTAC (proteolysis-targeting chimera) with Kd of 34 nM, 4.7 nM, 8.3 nM, 7.6 nM, 9.6 nM, and 7.6 nM for BRD2 (1), BRD2 (2), BRD3 (1), BRD3 (2), BRD4 (1), and BRD4 (2), respectively.
3 years -20°C powder
Beschrijving
ARV-771 Beschikbaar in 1 mg. Bestel eenvoudig online met snelle levering.
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