
Danusertib (PHA-739358)
Kwaliteit
ISO Gecertificeerd
Levering
24-48 uur
Technische Specificaties
827318-97-8
C07524-5mg
Aurora Kinase
Cell Cycle
CN1CCN (CC1) C2=CC=C (C=C2) C (=O) NC3=NNC4=C3CN (C4) C (=O) C (C5=CC=CC=C5) OC
C26H30N6O3
Danusertib (PHA-739358) is an Aurora kinase inhibitor for Aurora A/B/C with IC50 of 13 nM/79 nM/61 nM in cell-free assays, modestly potent to Abl, TrkA, c-RET and FGFR1, and less potent to Lck, VEGFR2/3, c-Kit, CDK2, etc. Danusertib induces apoptosis, cell cycle arrest, and autophagy. Phase 2.
2 years -80 in solvent
Beschrijving
Danusertib (PHA-739358) Beschikbaar in 5 mg. Wordt geleverd met droogijs. Bestel eenvoudig online met snelle levering.
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