Ensifentine
Gecertificeerd

Ensifentine

Catalog #: C14704-01
Maat: 5 mg

Kwaliteit

ISO Gecertificeerd

Levering

24-48 uur

Prijs -1%
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Gratis verzending vanaf €100

Technische Specificaties

CAS Number

1884461-72-6

Synonyms

RPL-554

SKU

C14704-5mg

Target

PDE

Applications

Metabolism

Molecular Formula

C26H31N5O4

Additionnal Information

Ensifentrine (RPL-554) is a first-in-class dual inhibitor of phosphodiesterase 3 (PDE3) and PDE4 with IC50 values of 0.4 nM and 1479 nM, respectively. Ensifentrine also inhibits lipopolysaccharide-induced tumor necrosis factor alpha release from human monocytes in a concentration-dependent manner. Ensifentrine demonstrates bronchoprotective and anti-inflammatory activities and can be used for chronic obstructive pulmonary disease (COPD) research.

Beschrijving

Ensifentine Beschikbaar in 5 mg. Bestel eenvoudig online met snelle levering.

Specificaties

ProductnaamEnsifentine
Categorie
Beschikbare grootte5 mg
CatalogusnummerC14704-01