GNE-781
Gecertificeerd

GNE-781

Catalog #: C13573-01
Maat: 5 mg

Kwaliteit

ISO Gecertificeerd

Levering

24-48 uur

Prijs -1%
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Gratis verzending vanaf €100

Technische Specificaties

CAS Number

1936422-33-1

SKU

C13573-5mg

Target

Epigenetic Reader Domain

Applications

Epigenetics

Smiles

CNC (=O) N1CCC2=C (C1) C (=N[N]2C3CCOCC3) N4CCCC5=C4C=C (C (F) F) C (=C5) C6=C[N] (C) N=C6

Molecular Formula

C27H33F2N7O2

Additionnal Information

GNE-781 (compound 19) is an orally active, highly potent and selective bromodomain inhibitor of cyclic adenosine monophosphate response element binding protein (CBP) with IC50 of 0.94 nM in TR-FRET assay. GNE-781 also inhibits BRET and BRD4 (1) with IC50 of 6.2 nM and 5100 nM, respectively. GNE-781 exhibits antitumor activity.

Storage Conditions

3 years -20°C powder

Beschrijving

GNE-781 Beschikbaar in 5 mg. Bestel eenvoudig online met snelle levering.

Specificaties

ProductnaamGNE-781
Categorie
Beschikbare grootte5 mg
CatalogusnummerC13573-01