S9-CMC1 TFA
Gecertificeerd

S9-CMC1 TFA

Catalog #: TP3001-01
Maat: 10 mg

Kwaliteit

ISO Gecertificeerd

Levering

24-48 uur

Prijs -1%
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BTW niet inbegrepen
Gratis verzending vanaf €100
Technische Documentatie

Technische Specificaties

Target

Apoptosis, Histone Demethylase

Related Pathways

Apoptosis, Chromatin/Epigenetic

Bioactivity

S9-CMC1 TFA is a covalent peptide lysine-specific demethylase 1 (LSD1) inhibitor with an IC50 value of 2.53 μM. It selectively targets the active site Cys360 of the enzyme. By inhibiting LSD1 activity, S9-CMC1 TFA elevates H3K4me1 and H3K4me2 levels, inducing G1 cell cycle arrest and apoptosis, thereby suppressing cell proliferation. In addition, S9-CMC1 TFA markedly inhibits tumor growth in A549 xenograft animal models.

Molecular Formula

C97H151F3N32O17S2

Molecular Weight

2158.57

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Beschrijving

S9-CMC1 TFA Beschikbaar in 10 mg. Bestel eenvoudig online met snelle levering.

Specificaties

ProductnaamS9-CMC1 TFA
Categorie
Beschikbare grootte10 mg
CatalogusnummerTP3001-01