
SRX3177
Kwaliteit
ISO Gecertificeerd
Levering
24-48 uur
Technische Specificaties
2241237-51-2
CDK
Cell Cycle
C31H32N6O4S
SRX3177 is a potent triple inhibitor targeting CDK4/6, PI3K, and BRD4, with IC50 values of 33 nM for BRD4 BD1, 89 nM for BRD4 BD2, 79 nM for PI3Kα, 83 nM for PI3Kδ, 3.18 μM for PI3Kγ, <2.5 nM for CDK4, and 3.3 nM for CDK6. By simultaneously inhibiting these key pathways, SRX3177 disrupts cancer cell signalling and exhibits significant cytotoxic effects in tumors.
Beschrijving
SRX3177 Beschikbaar in 25 mg. Bestel eenvoudig online met snelle levering.
Specificaties
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