Sulfated sulfakinine

Sulfated sulfakinin is a Sulfakinin receptor (SKR) activator with EC50s of 1.6 and 5.4 nM for Tribolium castaneumTc TcSKR1 and TcSKR2, respectively. SKRs are G-protein-coupled receptors (GPCRs) that interact with sulfakinins to modulate diverse biological processes. Sulfated sulfakinin can be used for tho control of pest insects research[1].

172430-35-2

12352209

Parasite

Anti-infection

Infection

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C54H71N15O17S2

1266.36

[1]Yu N, et al. Development of cell-based bioassay with Sf9 cells expressing TcSKR1 and TcSKR2 and differential activation by sulfated and non-sulfated SK peptides. Peptides. 2014 Mar;53:238-42.ptides.

Room temperature

http://file.medchemexpress.com/batch_PDF/HY-P11156/

Peptides

No Development Reported