TAT-CBD3A6K

1505463-57-9

Calcium Channel

Metabolism, Membrane transporter/Ion channel

TAT-CBD3A6K is a modified TAT-CBD3 peptide. It reduces T-type and R-type voltage-dependent calcium currents in dorsal root ganglion (DRG) neurons. By inhibiting CRMP-2-mediated enhancement of T-type and R-type calcium channel function, TAT-CBD3A6K exhibits anti-nociceptive effects in models of AIDS-induced peripheral neuropathy.

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C137H250N60O32

3249.83

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