WH-4-023
Gecertificeerd

WH-4-023

Catalog #: C17986
Maat: 100 mg
Droogijs Vereist

Kwaliteit

ISO Gecertificeerd

Levering

24-48 uur

Prijs -1%
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Gratis verzending vanaf €100

Technische Specificaties

CAS Number

837422-57-8

Synonyms

KIN001-112, KIN112, Dual LCK/SRC inhibitor

SKU

C17986-100mg

Target

Src

Applications

Protein Tyrosine Kinase

Smiles

CC1=C (C (=CC=C1) C) OC (=O) N (C2=C (C=C (C=C2) OC) OC) C3=NC (=NC=C3) NC4=CC=C (C=C4) N5CCN (CC5) C

Molecular Formula

C32H36N6O4

Additionnal Information

WH-4-023 (KIN001-112, KIN112, Dual LCK/SRC inhibitor) is a potent and orally active Lck/Src inhibitor with IC50s of 2 nM and 6 nM in cell-free assays, respectively. Exhibits >300-fold selectivity against p38α and KDR. Also potently inhibits SIK (IC50 values are 10, 22 and 60 nM for SIK 1, 2 and 3 respectively) and displays selectivity over a range of closely related kinases.

Storage Conditions

2 years -80 in solvent

Beschrijving

WH-4-023 Beschikbaar in 100 mg. Wordt geleverd met droogijs. Bestel eenvoudig online met snelle levering.

Specificaties

ProductnaamWH-4-023
Categorie
Beschikbare grootte100 mg
CatalogusnummerC17986